Publications
Aranda-Garcia, David and Stepniewski, Tomasz Maciej and Torrens-Fontanals, Mariona and Garcia-Recio, Adrian and Lopez-Balastegui, Marta and Medel-Lacruz, Brian and Morales-Pastor, Adrian and Peralta-Garcia, Alejandro and Dieguez-Eceolaza, Miguel and Sotillo-Nunez, David and Ding, Tianyi and Drabek, Matthaus and Jacquemard, Celien and Jakowiecki, Jakub and Jespers, Willem and Jimenez-Roses, Mireia and Jun-Yu-Lim, Victor and Nicoli, Alessandro and Orzel, Urszula and Shahraki, Aida and Tiemann, Johanna K. S. and Ledesma-Martin, Vicente and Nerin-Fonz, Francho and Suarez-Dou, Sergio and Canal, Oriol and Pandy-Szekeres, Gaspar and Mao, Jiafei and Gloriam, David E. and Kellenberger, Esther and Latek, Dorota and Guixa-Gonzalez, Ramon and Gutierrez-de-Teran, Hugo and Tikhonova, Irina G. and Hildebrand, Peter W. and Filizola, Marta and Babu, M. Madan and Di Pizio, Antonella and Filipek, Slawomir and Kolb, Peter and Cordomi, Arnau and Giorgino, Toni and Marti-Solano, Maria and Selent, Jana. 2025. Large scale investigation of GPCR molecular dynamics data uncovers allosteric sites and lateral gateways. Nature Communications 16 (1). doi: 10.1038/s41467-025-57034-y. (http://dx.doi.org/10.1038/s41467-025-57034-y)
Dynamic id | Receptor | Model name | Uniprot entry name | Uniprot ID | Family | Class | PDB ID | State | Species | Model type | Source type | Ligand(s) | Num. of atoms | Membrane composition | Accum. sim. time (µs) | Software | Force field | Submitted by | ||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
View | 909 | 5-hydroxytryptamine receptor 1b | 5-hydroxytryptamine receptor 1b in complex with RLJFTICUTY... | 5ht1b_human | P28222 | 5-Hydroxytryptamine receptors | A | 5V54 | Inactive | Homo sapiens | Complex | X-ray | Chembl428892 | 75470 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 908 | 5-hydroxytryptamine receptor 1b | 5-hydroxytryptamine receptor 1b (apoform) | 5ht1b_human | P28222 | 5-Hydroxytryptamine receptors | A | 5V54 | Inactive | Homo sapiens | Apoform | X-ray | 75414 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 802 | 5-hydroxytryptamine receptor 2a | 5-hydroxytryptamine receptor 2a in complex with HDOZVRUNCM... | 5ht2a_human | P28223 | 5-Hydroxytryptamine receptors | A | 6A94 | Inactive | Homo sapiens | Complex | X-ray | Zotepine | 59717 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 849 | 5-hydroxytryptamine receptor 2a | 5-hydroxytryptamine receptor 2a in complex with RAPZEAPATH... | 5ht2a_human | P28223 | 5-Hydroxytryptamine receptors | A | 6A93 | Inactive | Homo sapiens | Complex | X-ray | Risperidone | 83220 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 848 | 5-hydroxytryptamine receptor 2a | 5-hydroxytryptamine receptor 2a (apoform) | 5ht2a_human | P28223 | 5-Hydroxytryptamine receptors | A | 6A93 | Inactive | Homo sapiens | Apoform | X-ray | 83142 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 801 | 5-hydroxytryptamine receptor 2a | 5-hydroxytryptamine receptor 2a (apoform) | 5ht2a_human | P28223 | 5-Hydroxytryptamine receptors | A | 6A94 | Inactive | Homo sapiens | Apoform | X-ray | 59628 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 719 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor in complex with BKRGVLQUQGGVSM-KBXCAEBGSA-N | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DRX | Intermediate | Homo sapiens | Complex | X-ray | Arolac | 72108 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 812 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor in complex with KPJZHOPZRAFDTN-ZRGWGRIASA-N | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DRZ | Intermediate | Homo sapiens | Complex | X-ray | Metisergide | 78753 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 820 | 5-hydroxytryptamine receptor 2b | chimera protein of human 5-hydroxytryptamine receptor 2b a... | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 4NC3 | Intermediate | Homo sapiens | Complex | X-ray | Ergotamine | 69501 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 847 | 5-hydroxytryptamine receptor 2b | chimera protein of human 5-hydroxytryptamine receptor 2b a... | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 5TVN | Intermediate | Homo sapiens | Complex | X-ray | Haze | 80303 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 919 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor in complex with UNBRKDKAWYKMIV-QWQRMKEZSA-N | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DRY | Intermediate | Homo sapiens | Complex | X-ray | Methylergonovine | 79912 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 960 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor in complex with NJLHHCITDFZZSE-KRWDZBQOSA-N | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DS0 | Intermediate | Homo sapiens | Complex | X-ray | (1s)-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-6-methyl-2,3... | 68794 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 959 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor (apoform) | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DS0 | Intermediate | Homo sapiens | Apoform | X-ray | 68684 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 918 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor (apoform) | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DRY | Intermediate | Homo sapiens | Apoform | X-ray | 79801 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 846 | 5-hydroxytryptamine receptor 2b | chimera protein of human 5-hydroxytryptamine receptor 2b a... | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 5TVN | Intermediate | Homo sapiens | Apoform | X-ray | 80202 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 819 | 5-hydroxytryptamine receptor 2b | chimera protein of human 5-hydroxytryptamine receptor 2b a... | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 4NC3 | Intermediate | Homo sapiens | Apoform | X-ray | 69362 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 811 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor (apoform) | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DRZ | Intermediate | Homo sapiens | Apoform | X-ray | 78642 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 718 | 5-hydroxytryptamine receptor 2b | 5ht2b receptor (apoform) | 5ht2b_human | P41595 | 5-Hydroxytryptamine receptors | A | 6DRX | Intermediate | Homo sapiens | Apoform | X-ray | 71991 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 990 | Muscarinic acetylcholine receptor m2 | muscarinic acetylcholine receptor m2 in complex with HGMIT... | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZK3 | Inactive | Homo sapiens | Complex | X-ray | Quinuclidinyl benzilate | 109307 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1029 | Muscarinic acetylcholine receptor m2 | muscarinic acetylcholine receptor m2 in complex with MZDYA... | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZKB | Inactive | Homo sapiens | Complex | X-ray | Chembl1318307 | 66939 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1096 | Muscarinic acetylcholine receptor m2 | M2 muscarinic acetylcholine receptor in complex with NMS | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZK8 | Inactive | Homo sapiens | Complex | X-ray | Paminereg | 99783 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1126 | Muscarinic acetylcholine receptor m2 | M2 muscarinic acetylcholine receptor in complex with with... | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZKC | Inactive | Homo sapiens | Complex | X-ray | Paminereg | 95417 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1127 | Muscarinic acetylcholine receptor m2 | M2 muscarinic acetylcholine receptor bound with NMS | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5YC8 | Inactive | Homo sapiens | Complex | X-ray | Paminereg | 112748 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1122 | Muscarinic acetylcholine receptor m2 | M2 muscarinic acetylcholine receptor | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5YC8 | Inactive | Homo sapiens | Apoform | X-ray | 112707 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1028 | Muscarinic acetylcholine receptor m2 | muscarinic acetylcholine receptor m2 (apoform) | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZKB | Inactive | Homo sapiens | Apoform | X-ray | 100272 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 989 | Muscarinic acetylcholine receptor m2 | muscarinic acetylcholine receptor m2 (apoform) | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZK3 | Inactive | Homo sapiens | Apoform | X-ray | 99695 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 968 | Muscarinic acetylcholine receptor m2 | muscarinic acetylcholine receptor m2 (apoform) | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZKC | Inactive | Homo sapiens | Apoform | X-ray | 95404 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 797 | Muscarinic acetylcholine receptor m2 | muscarinic acetylcholine receptor m2 (apoform) | acm2_human | P08172 | Acetylcholine receptors (muscarinic) | A | 5ZK8 | Inactive | Homo sapiens | Apoform | X-ray | 99746 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1125 | Muscarinic acetylcholine receptor m3 | M3 muscarinic acetylcholine receptor in complex with a sel... | acm3_rat | P08483 | Acetylcholine receptors (muscarinic) | A | 5ZHP | Inactive | Rattus norvegicus | Complex | X-ray | Compound 34 | 62040 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 947 | Muscarinic acetylcholine receptor m3 | muscarinic acetylcholine receptor m3 (apoform) | acm3_rat | P08483 | Acetylcholine receptors (muscarinic) | A | 5ZHP | Inactive | Rattus norvegicus | Apoform | X-ray | 85097 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 983 | Muscarinic acetylcholine receptor m4 | muscarinic acetylcholine receptor m4 (apoform) | acm4_human | P08173 | Acetylcholine receptors (muscarinic) | A | 6KP6 | Inactive | Homo sapiens | Apoform | X-ray | 89925 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1094 | Muscarinic acetylcholine receptor m5 | M5 muscarinic acetylcholine receptor in complex with tiotr... | acm5_human | P08912 | Acetylcholine receptors (muscarinic) | A | 6OL9 | Inactive | Homo sapiens | Complex | X-ray | Tiotropium | 64844 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 973 | Muscarinic acetylcholine receptor m5 | muscarinic acetylcholine receptor m5 (apoform) | acm5_human | P08912 | Acetylcholine receptors (muscarinic) | A | 6OL9 | Inactive | Homo sapiens | Apoform | X-ray | 91509 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 729 | Beta-1 adrenergic receptor | beta-1 adrenergic receptor in complex with CQEFAUFOQSCRMZ-... | adrb1_melga | P07700 | Adrenoceptors | A | 5F8U | Inactive | Meleagris gallopavo | Complex | X-ray | 4-{[(2s)-3-(tert-butylamino)-2-hydroxypropyl]oxy}-3h-indol... | 92001 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 786 | Beta-1 adrenergic receptor | beta-1 adrenergic receptor in complex with JBLUMBNIBNHRSO-... | adrb1_melga | P07700 | Adrenoceptors | A | 2YCZ | Inactive | Meleagris gallopavo | Complex | X-ray | 4-{[(2s)-3-(tert-butylamino)-2-hydroxypropyl]oxy}-3-iodo-1... | 92017 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 961 | Beta-1 adrenergic receptor | beta-1 adrenergic receptor (apoform) | adrb1_melga | P07700 | Adrenoceptors | A | 4GPO | Inactive | Meleagris gallopavo | Apoform | X-ray | 96570 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 785 | Beta-1 adrenergic receptor | beta-1 adrenergic receptor (apoform) | adrb1_melga | P07700 | Adrenoceptors | A | 2YCZ | Inactive | Meleagris gallopavo | Apoform | X-ray | 91980 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 728 | Beta-1 adrenergic receptor | beta-1 adrenergic receptor (apoform) | adrb1_melga | P07700 | Adrenoceptors | A | 5F8U | Inactive | Meleagris gallopavo | Apoform | X-ray | 85204 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 685 | Beta-2 adrenergic receptor | 6PS0 complex | adrb2_human | P07550 | Adrenoceptors | A | 6PS0 | Inactive | Homo sapiens | Complex | X-ray | (s)-carazolol | None | CLR POPC | 0.15 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 752 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS5 | Inactive | Homo sapiens | Complex | X-ray | Chembl452861 | 91650 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 764 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS1 | Inactive | Homo sapiens | Complex | X-ray | Aquanil | 94398 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 770 | Beta-2 adrenergic receptor | chimera protein of beta-2 adrenergic receptor and lysozyme... | adrb2_human | P07550 | Adrenoceptors | A | 5X7D | Inactive | Homo sapiens | Complex | X-ray | (s)-carazolol | 96671 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 830 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS4 | Inactive | Homo sapiens | Complex | X-ray | Chembl1233766 | 94382 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 864 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS2 | Inactive | Homo sapiens | Complex | X-ray | (-)-alprenolol | 89928 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 927 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS3 | Inactive | Homo sapiens | Complex | X-ray | (s)-carvedilol | 95741 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 952 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS6 | Inactive | Homo sapiens | Complex | X-ray | Aquanil | 92031 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 963 | Beta-2 adrenergic receptor | beta-2 adrenergic receptor in complex with BQXQGZPYHWWCEB-... | adrb2_human | P07550 | Adrenoceptors | A | 5D6L | Inactive | Homo sapiens | Complex | X-ray | (s)-carazolol | 88157 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 971 | Beta-2 adrenergic receptor | beta-2 adrenergic receptor in complex with BQXQGZPYHWWCEB-... | adrb2_human | P07550 | Adrenoceptors | A | 4GBR | Inactive | Homo sapiens | Complex | X-ray | (s)-carazolol | 84422 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 980 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PRZ | Inactive | Homo sapiens | Complex | X-ray | (-)-alprenolol | 91905 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1130 | Beta-2 adrenergic receptor | beta-2 adrenergic receptor in complex with 6-bromo-N~2~-ph... | adrb2_human | P07550 | Adrenoceptors | A | 6OBA | Inactive | Homo sapiens | Complex | X-ray | (-)-alprenolol 6-bromo-n~2~-phenylquinazoline-2,4-diamine | 94583 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 829 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS4 | Inactive | Homo sapiens | Apoform | X-ray | 94281 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 763 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS1 | Inactive | Homo sapiens | Apoform | X-ray | 94299 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1003 | Beta-2 adrenergic receptor | beta-2 adrenergic receptor (apoform) | adrb2_human | P07550 | Adrenoceptors | A | 6OBA | Inactive | Homo sapiens | Apoform | X-ray | 94468 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 979 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PRZ | Inactive | Homo sapiens | Apoform | X-ray | 91816 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 970 | Beta-2 adrenergic receptor | beta-2 adrenergic receptor (apoform) | adrb2_human | P07550 | Adrenoceptors | A | 4GBR | Inactive | Homo sapiens | Apoform | X-ray | 84374 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 962 | Beta-2 adrenergic receptor | beta-2 adrenergic receptor (apoform) | adrb2_human | P07550 | Adrenoceptors | A | 5D6L | Inactive | Homo sapiens | Apoform | X-ray | 88024 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 951 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS6 | Inactive | Homo sapiens | Apoform | X-ray | 91938 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 926 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS3 | Inactive | Homo sapiens | Apoform | X-ray | 95628 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 863 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS2 | Inactive | Homo sapiens | Apoform | X-ray | 89833 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 769 | Beta-2 adrenergic receptor | chimera protein of beta-2 adrenergic receptor and lysozyme... | adrb2_human | P07550 | Adrenoceptors | A | 5X7D | Inactive | Homo sapiens | Apoform | X-ray | 96474 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 751 | Beta-2 adrenergic receptor | fusion protein of beta-2 adrenergic receptor and t4 lysozy... | adrb2_human | P07550 | Adrenoceptors | A | 6PS5 | Inactive | Homo sapiens | Apoform | X-ray | 91553 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 684 | Beta-2 adrenergic receptor | 6PS0 apoform | adrb2_human | P07550 | Adrenoceptors | A | 6PS0 | Inactive | Homo sapiens | Apoform | X-ray | None | POPC | 0.15 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 839 | D(2) dopamine receptor | chimera of d(2) dopamine receptor and endolysin in complex... | drd2_human | P14416 | Dopamine receptors | A | 6LUQ | Inactive | synthetic | Complex | X-ray | Aloperidolo | 94255 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 925 | D(2) dopamine receptor | d(2) dopamine receptor in complex with RAPZEAPATHNIPO-UHFF... | drd2_human | P14416 | Dopamine receptors | A | 6CM4 | Inactive | synthetic | Complex | X-ray | Risperidone | 82215 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 924 | D(2) dopamine receptor | d(2) dopamine receptor (apoform) | drd2_human | P14416 | Dopamine receptors | A | 6CM4 | Inactive | Homo sapiens | Apoform | X-ray | 82152 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 838 | D(2) dopamine receptor | chimera of d(2) dopamine receptor and endolysin (apoform) | drd2_human | P14416 | Dopamine receptors | A | 6LUQ | Inactive | Homo sapiens | Apoform | X-ray | 94201 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 832 | D(4) dopamine receptor | d(4) dopamine receptor in complex with Nemonapride | drd4_human | P21917 | Dopamine receptors | A | 5WIV | Inactive | Homo sapiens | Complex | X-ray | Nemonapride | 90817 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1006 | D(4) dopamine receptor | d(4) dopamine receptor in complex with Nemonapride | drd4_human | P21917 | Dopamine receptors | A | 5WIU | Inactive | Homo sapiens | Complex | X-ray | Nemonapride | 75922 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1005 | D(4) dopamine receptor | d(4) dopamine receptor (apoform) | drd4_human | P21917 | Dopamine receptors | A | 5WIU | Inactive | Homo sapiens | Apoform | X-ray | 75866 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 831 | D(4) dopamine receptor | d(4) dopamine receptor (apoform) | drd4_human | P21917 | Dopamine receptors | A | 5WIV | Inactive | Homo sapiens | Apoform | X-ray | 90758 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 891 | Type-2 angiotensin ii receptor | chimera protein of type-2 angiotensin ii receptor and solu... | agtr2_human | P50052 | Angiotensin receptors | A | 5UNG | Active | Homo sapiens | Complex | X-ray | Chembl289472 | 74483 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 917 | Type-2 angiotensin ii receptor | chimera protein of type-2 angiotensin ii receptor and solu... | agtr2_human | P50052 | Angiotensin receptors | A | 5UNF | Active | Homo sapiens | Complex | X-ray | Chembl289472 | 69129 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 940 | Type-2 angiotensin ii receptor | type-2 angiotensin ii receptor in complex with SYDVEZUPFQX... | agtr2_human | P50052 | Angiotensin receptors | A | 5UNH | Active | Homo sapiens | Complex | X-ray | N-[(furan-2-yl)methyl]-n-(4-oxo-2-propyl-3-{[2'-(2h-tetraz... | 69317 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 939 | Type-2 angiotensin ii receptor | type-2 angiotensin ii receptor (apoform) | agtr2_human | P50052 | Angiotensin receptors | A | 5UNH | Active | Homo sapiens | Apoform | X-ray | 69239 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 916 | Type-2 angiotensin ii receptor | chimera protein of type-2 angiotensin ii receptor and solu... | agtr2_human | P50052 | Angiotensin receptors | A | 5UNF | Active | Homo sapiens | Apoform | X-ray | 69052 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 890 | Type-2 angiotensin ii receptor | chimera protein of type-2 angiotensin ii receptor and solu... | agtr2_human | P50052 | Angiotensin receptors | A | 5UNG | Active | Homo sapiens | Apoform | X-ray | 74403 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1062 | Apelin receptor | Apelin receptor in complex with agonist peptide | apj_human | P35414 | Apelin receptors | A | 5VBL | Inactive | Homo sapiens | Complex | X-ray | 78954 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1042 | Apelin receptor | Apelin receptor in complex with single domain antibody JN241 | apj_human | - P35414 | Apelin receptors | A | 6KNM | Inactive | Homo sapiens | Complex | X-ray | Single domain antibody jn241 | 123845 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1041 | Apelin receptor | Apelin receptor (apoform) | apj_human | P35414 | Apelin receptors | A | 6KNM | Inactive | Homo sapiens | Apoform | X-ray | 92450 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1063 | Apelin receptor | Apelin receptor (apoform) | apj_human | P35414 | Apelin receptors | A | 5VBL | Inactive | Homo sapiens | Apoform | X-ray | 78954 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 921 | C5a anaphylatoxin chemotactic receptor 1 | c5a anaphylatoxin chemotactic receptor 1 in complex with I... | c5ar1_human | P21730 | Complement peptide receptors | A | 5O9H | Inactive | Homo sapiens | Complex | X-ray | Chembl4303272 | 64894 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1100 | C5a anaphylatoxin chemotactic receptor 1 | 6C1R in complex with PMX53 | c5ar1_human | P21730 | Complement peptide receptors | A | 6C1R | Inactive | Homo sapiens | Complex | X-ray | Avacopan | 68210 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1131 | C5a anaphylatoxin chemotactic receptor 1 | C5a receptor in complex with an orthosteric antagonist PMX... | c5ar1_human | P21730 | Complement peptide receptors | A | 6C1Q | Inactive | Homo sapiens | Complex | X-ray | Chembl4303272 | 66982 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1085 | C5a anaphylatoxin chemotactic receptor 1 | 6C1R apoform | c5ar1_human | P21730 | Complement peptide receptors | A | 6C1R | Inactive | Homo sapiens | Apoform | X-ray | 66801 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1084 | C5a anaphylatoxin chemotactic receptor 1 | 6C1Q apoform | c5ar1_human | P21730 | Complement peptide receptors | A | 6C1Q | Inactive | Homo sapiens | Apoform | X-ray | 66801 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 920 | C5a anaphylatoxin chemotactic receptor 1 | c5a anaphylatoxin chemotactic receptor 1 (apoform) | c5ar1_human | P21730 | Complement peptide receptors | A | 5O9H | Inactive | Homo sapiens | Apoform | X-ray | 64943 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 788 | Endothelin b receptor | endothelin b receptor in complex with UZDORQWMYRRLQV-JHOUS... | ednrb_human | P24530 | Endothelin receptors | A | 6K1Q | Inactive | Homo sapiens | Complex | X-ray | Chembl72410 | 91505 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 887 | Endothelin b receptor | endothelin b receptor in complex with GJPICJJJRGTNOD-UHFFF... | ednrb_human | P24530 | Endothelin receptors | A | 5XPR | Inactive | Homo sapiens | Complex | X-ray | Actelion | 90331 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 965 | Endothelin b receptor | endothelin b receptor in complex with MTNFANNLCUMCNB-UHFFF... | ednrb_human | P24530 | Endothelin receptors | A | 5X93 | Inactive | Homo sapiens | Complex | X-ray | 3-[6-[(4-tert-butylphenyl)sulfonylamino]-5-(2-methoxypheno... | 84641 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1016 | Endothelin b receptor | endothelin receptor type b in complex with endothelin-3 | ednrb_human | P24530 | Endothelin receptors | A | 6IGK | Inactive | Homo sapiens | Complex | X-ray | 76115 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1064 | Endothelin b receptor | Endothelin receptor type B in complex with IRL 1620 | ednrb_human | P24530 | Endothelin receptors | A | 6IGL | Inactive | Homo sapiens | Complex | X-ray | 97624 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 997 | Sarafotoxin [cleaved into: sarafotoxin-a, ser-isoform | endothelin receptor type b in complex with sarafotoxin-b | ednrb_human | P24530 P13208 | None | A | 6LRY | Inactive | Atractaspis engaddensis | Complex | X-ray | Sarafotoxin [cleaved into: sarafotoxin-a, ser-isoform | 82288 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 837 | Endothelin receptor type b | endothelin receptor subtype-b (apoform) | ednrb_human | P24530 | Endothelin receptors | A | 5GLI | Inactive | Homo sapiens | Apoform | X-ray | 82661 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 787 | Endothelin receptor type b | endothelin b receptor (apoform) | ednrb_human | P24530 | Endothelin receptors | A | 6K1Q | Inactive | Homo sapiens | Apoform | X-ray | 91424 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1059 | Endothelin receptor type b | Endothelin receptor type B (apoform) | ednrb_human | P24530 | Endothelin receptors | A | 6IGL | Inactive | Homo sapiens | Apoform | X-ray | 97352 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1015 | Endothelin receptor type b | endothelin receptor type b (apoform) | ednrb_human | P24530 | Endothelin receptors | A | 6IGK | Inactive | Homo sapiens | Apoform | X-ray | 75902 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 996 | Endothelin receptor type b | endothelin receptor type b (apoform) | ednrb_human | P24530 | Endothelin receptors | A | 6LRY | Inactive | Homo sapiens | Apoform | X-ray | 82107 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 964 | Endothelin receptor type b | endothelin b receptor (apoform) | ednrb_human | P24530 | Endothelin receptors | A | 5X93 | Inactive | Homo sapiens | Apoform | X-ray | 84520 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 886 | Endothelin receptor type b | endothelin b receptor (apoform) | ednrb_human | P24530 | Endothelin receptors | A | 5XPR | Inactive | Homo sapiens | Apoform | X-ray | 90264 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1081 | N-formyl peptide receptor 2 | 6LW5 in complex with WKYMVm | fpr2_human | P25090 | Formylpeptide receptors | A | 6LW5 | Active | Homo sapiens | Complex | X-ray | D-methioninamide | 71197 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1082 | N-formyl peptide receptor 2 | 6LW5 apoform | fpr2_human | P25090 | Formylpeptide receptors | A | 6LW5 | Active | Homo sapiens | Apoform | X-ray | 69420 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 905 | Neuropeptide y receptor type 1 | neuropeptide y receptor type 1 in complex with WMYSXJSJXZF... | npy1r_human | P25929 | Neuropeptide Y receptors | A | 5ZBH | Inactive | Homo sapiens | Complex | X-ray | 3,5-pyridinedicarboxylic acid, 1,4-dihydro-4-(3-((((3-(4-(... | 80434 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1040 | Neuropeptide y receptor type 1 | neuropeptide y receptor type 1 in complex with VQHNWOOVOKY... | npy1r_human | P25929 | Neuropeptide Y receptors | A | 5ZBQ | Inactive | Homo sapiens | Complex | X-ray | Chembl3747822 | 81605 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 700 | Neuropeptide y receptor type 1 | neuropeptide y receptor type 1 (apoform) | npy1r_human | P25929 | Neuropeptide Y receptors | A | 5ZBQ | Inactive | Homo sapiens | Apoform | X-ray | 81522 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 904 | Neuropeptide y receptor type 1 | neuropeptide y receptor type 1 (apoform) | npy1r_human | P25929 | Neuropeptide Y receptors | A | 5ZBH | Inactive | Homo sapiens | Apoform | X-ray | 80351 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 723 | Neurotensin receptor type 1 | neurotensin receptor type 1 in complex with arg-arg-pro-ty... | ntr1_rat | P20789 | Neurotensin receptors | A | 5T04 | Active | Rattus norvegicus | Complex | X-ray | 90561 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 768 | Neurotensin receptor type 1 | neurotensin receptor type 1 in complex with neurotensin/ne... | ntr1_rat | P20789 | Neurotensin receptors | A | 4XES | Active | Rattus norvegicus | Complex | X-ray | 87947 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 881 | Neurotensin receptor type 1 | neurotensin receptor type 1 in complex with GLYCINE | ntr1_rat | P20789 | Neurotensin receptors | A | 4BUO | Inactive | Rattus norvegicus | Complex | X-ray | Glycine | 89811 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 767 | Neurotensin receptor type 1 | neurotensin receptor type 1 (apoform) | ntr1_rat | P20789 | Neurotensin receptors | A | 4XES | Active | Rattus norvegicus | Apoform | X-ray | 87822 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 880 | Neurotensin receptor type 1 | neurotensin receptor type 1 (apoform) | ntr1_rat | P20789 | Neurotensin receptors | A | 4BUO | Inactive | Rattus norvegicus | Apoform | X-ray | 89606 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 722 | Neurotensin receptor type 1 | neurotensin receptor type 1 (apoform) | ntr1_rat | P20789 | Neurotensin receptors | A | 5T04 | Active | Rattus norvegicus | Apoform | X-ray | 90469 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 725 | Delta-type opioid receptor | delta-type opioid receptor in complex with WIYUZYBFCWCCQJ-... | oprd_mouse | P32300 | Opioid receptors | A | 4EJ4 | Inactive | Mus musculus | Complex | X-ray | Naltrindole | 79548 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 724 | Delta-type opioid receptor | delta-type opioid receptor (apoform) | oprd_mouse | P32300 | Opioid receptors | A | 4EJ4 | Inactive | Mus musculus | Apoform | X-ray | 79281 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 737 | Orexin receptor type 1 | orexin receptor type 1 in complex with AKMNUCBQGHFICM-UHFF... | ox1r_human | O43613 | Orexin receptors | A | 6TQ7 | Inactive | Homo sapiens | Complex | X-ray | Chembl291536 | 91907 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 760 | Orexin receptor type 1 | orexin receptor type 1 in complex with NHPQGZOBHSVTAQ-IBGZ... | ox1r_human | O43613 | Orexin receptors | A | 6TP4 | Inactive | Homo sapiens | Complex | X-ray | Chembl3597952 | 93728 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 822 | Orexin receptor type 1 | orexin receptor type 1 in complex with TWCRHJLMMAYSTE-ZFWW... | ox1r_human | O43613 | Orexin receptors | A | 6TOS | Inactive | Homo sapiens | Complex | X-ray | Chembl2413522 | 86031 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 834 | Orexin receptor type 1 | orexin receptor type 1 in complex with JTARFZSNUAGHRB-UHFF... | ox1r_human | O43613 | Orexin receptors | A | 6TQ9 | Inactive | Homo sapiens | Complex | X-ray | Ac1n7qoy | 91799 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 860 | Orexin receptor type 1 | orexin receptor type 1 in complex with LWKUASRJTUZHSJ-UHFF... | ox1r_human | O43613 | Orexin receptors | A | 6TQ6 | Inactive | Homo sapiens | Complex | X-ray | Chembl4592653 | 89637 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 870 | Orexin receptor type 1 | orexin receptor type 1 in complex with NPFDWHQSDBWQLH-QZTJ... | ox1r_human | O43613 | Orexin receptors | A | 6TP6 | Inactive | Homo sapiens | Complex | X-ray | Filorexant | 91312 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 875 | Orexin receptor type 1 | orexin receptor type 1 in complex with MUGXRYIUWFITCP-PGRD... | ox1r_human | O43613 | Orexin receptors | A | 6TOT | Inactive | Homo sapiens | Complex | X-ray | Lemborexant | 91689 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 915 | Orexin receptor type 1 | orexin receptor type 1 in complex with KJPHTXTWFHVJIG-UHFF... | ox1r_human | O43613 | Orexin receptors | A | 6TOD | Inactive | Homo sapiens | Complex | X-ray | Empa | 85638 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 936 | Orexin receptor type 1 | orexin receptor type 1 in complex with JYTNQNCOQXFQPK-MRXN... | ox1r_human | O43613 | Orexin receptors | A | 6TO7 | Inactive | Homo sapiens | Complex | X-ray | Suvorexant | 94091 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 967 | Orexin receptor type 1 | orexin receptor type 1 in complex with KIKWLYIDCILHAP-UHFF... | ox1r_human | O43613 | Orexin receptors | A | 6TQ4 | Inactive | Homo sapiens | Complex | X-ray | Chembl4590386 | 94536 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 966 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TQ4 | Inactive | Homo sapiens | Apoform | X-ray | 94480 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 833 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TQ9 | Inactive | Homo sapiens | Apoform | X-ray | 91747 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 821 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TOS | Inactive | Homo sapiens | Apoform | X-ray | 85982 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 758 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TP3 | Inactive | Homo sapiens | Apoform | X-ray | 98232 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 935 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TO7 | Inactive | Homo sapiens | Apoform | X-ray | 94004 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 914 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TOD | Inactive | Homo sapiens | Apoform | X-ray | 85620 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 874 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TOT | Inactive | Homo sapiens | Apoform | X-ray | 91656 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 869 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TP6 | Inactive | Homo sapiens | Apoform | X-ray | 91248 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 859 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TQ6 | Inactive | Homo sapiens | Apoform | X-ray | 89459 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 759 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TP4 | Inactive | Homo sapiens | Apoform | X-ray | 93694 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 736 | Orexin/hypocretin receptor type 1 | orexin receptor type 1 (apoform) | ox1r_human | O43613 | Orexin receptors | A | 6TQ7 | Inactive | Homo sapiens | Apoform | X-ray | 91830 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 727 | Orexin receptor type 2 | orexin receptor type 2 in complex with KJPHTXTWFHVJIG-UHFF... | ox2r_human | O43614 | Orexin receptors | A | 5WS3 | Inactive | Homo sapiens | Complex | X-ray | Empa | 103282 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 745 | Orexin receptor type 2 | hypocretin receptor-2 in complex with JYTNQNCOQXFQPK-MRXNP... | ox2r_human | O43614 | Orexin receptors | A | 6TPJ | Inactive | Homo sapiens | Complex | X-ray | Suvorexant | 104023 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 845 | Orexin receptor type 2 | orexin receptor type 2 in complex with KJPHTXTWFHVJIG-UHFF... | ox2r_human | O43614 | Orexin receptors | A | 5WQC | Inactive | Homo sapiens | Complex | X-ray | Empa | 96313 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 866 | Orexin receptor type 2 | hypocretin receptor-2 in complex with KJPHTXTWFHVJIG-UHFFF... | ox2r_human | O43614 | Orexin receptors | A | 6TPG | Inactive | Homo sapiens | Complex | X-ray | Empa | 92750 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 903 | Orexin receptor type 2 | orexin receptor type 2 in complex with SUQZCEUKWPKXEE-UHFF... | ox2r_human | O43614 | Orexin receptors | A | 6TPN | Inactive | Homo sapiens | Complex | X-ray | Chembl3740099 | 93248 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 844 | Orexin receptor type 2 | orexin receptor type 2 (apoform) | ox2r_human | O43614 | Orexin receptors | A | 5WQC | Inactive | Homo sapiens | Apoform | X-ray | 96247 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 902 | Orexin receptor type 2 | orexin receptor type 2 (apoform) | ox2r_human | O43614 | Orexin receptors | A | 6TPN | Inactive | Homo sapiens | Apoform | X-ray | 93201 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 865 | Orexin receptor type 2 | hypocretin receptor-2 (apoform) | ox2r_human | O43614 | Orexin receptors | A | 6TPG | Inactive | Homo sapiens | Apoform | X-ray | 92693 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 744 | Orexin receptor type 2 | hypocretin receptor-2 (apoform) | ox2r_human | O43614 | Orexin receptors | A | 6TPJ | Inactive | Homo sapiens | Apoform | X-ray | 103972 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 726 | Orexin receptor type 2 | orexin receptor type 2 (apoform) | ox2r_human | O43614 | Orexin receptors | A | 5WS3 | Inactive | Homo sapiens | Apoform | X-ray | 103216 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 978 | Proteinase-activated receptor 2 | proteinase-activated receptor 2 in complex with IDFPQEHZYB... | par2_human | P55085 | Proteinase-activated receptors | A | 5NDD | Active | Homo sapiens | Complex | X-ray | Chembl4127372 | 78210 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1019 | Proteinase-activated receptor 2 | proteinase-activated receptor 2 in complex with FJAOGFGHTP... | par2_human | P55085 | Proteinase-activated receptors | A | 5NDZ | Active | Homo sapiens | Complex | X-ray | Chembl4128763 | 75018 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 977 | Proteinase-activated receptor 2 | proteinase-activated receptor 2 (apoform) | par2_human | P55085 | Proteinase-activated receptors | A | 5NDD | Active | Homo sapiens | Apoform | X-ray | 78178 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1018 | Proteinase-activated receptor 2 | proteinase-activated receptor 2 (apoform) | par2_human | P55085 | Proteinase-activated receptors | A | 5NDZ | Active | Homo sapiens | Apoform | X-ray | 74960 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 731 | Substance-p receptor | substance-p receptor in complex with ATALOFNDEOCMKK-OITMNO... | nk1r_human | P25103 | Tachykinin receptors | A | 6HLO | Inactive | Homo sapiens | Complex | X-ray | Cid 6918365 | 76114 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 782 | Substance-p receptor | substance-p receptor in complex with ATALOFNDEOCMKK-OITMNO... | nk1r_human | P25103 | Tachykinin receptors | A | 6J21 | Inactive | Homo sapiens | Complex | X-ray | Cid 6918365 | 79631 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 851 | Substance-p receptor | substance-p receptor in complex with DTQNEFOKTXXQKV-HKUYNN... | nk1r_human | P25103 | Tachykinin receptors | A | 6HLL | Inactive | Homo sapiens | Complex | X-ray | Chembl441225 | 81122 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 856 | Substance-p receptor | substance-p receptor chimera in complex with USRYEHHMJIRI... | nk1r_human | P25103 | Tachykinin receptors | A | 6E59 | Inactive | Homo sapiens | Complex | X-ray | Chembl4303434 | 86290 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 911 | Substance-p receptor | substance-p receptor in complex with ATALOFNDEOCMKK-OITMNO... | nk1r_human | P25103 | Tachykinin receptors | A | 6J20 | Inactive | Homo sapiens | Complex | X-ray | Cid 6918365 | 83214 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 938 | Substance-p receptor | substance-p receptor in complex with WAXQNWCZJDTGBU-UHFFFA... | nk1r_human | P25103 | Tachykinin receptors | A | 6HLP | Inactive | Homo sapiens | Complex | X-ray | Netupitant | 75351 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 781 | Substance-p receptor | substance-p receptor (apoform) | nk1r_human | P25103 | Tachykinin receptors | A | 6J21 | Inactive | Homo sapiens | Apoform | X-ray | 79574 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 937 | Substance-p receptor | substance-p receptor (apoform) | nk1r_human | P25103 | Tachykinin receptors | A | 6HLP | Inactive | Homo sapiens | Apoform | X-ray | 75280 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 910 | Substance-p receptor | substance-p receptor (apoform) | nk1r_human | P25103 | Tachykinin receptors | A | 6J20 | Inactive | Homo sapiens | Apoform | X-ray | 83157 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 855 | Substance-p receptor | substance-p receptor chimera (apoform) | nk1r_human | P25103 | Tachykinin receptors | A | 6E59 | Inactive | Homo sapiens | Apoform | X-ray | 84970 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 850 | Substance-p receptor | substance-p receptor (apoform) | nk1r_human | P25103 | Tachykinin receptors | A | 6HLL | Inactive | Homo sapiens | Apoform | X-ray | 81078 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 730 | Substance-p receptor | substance-p receptor (apoform) | nk1r_human | P25103 | Tachykinin receptors | A | 6HLO | Inactive | Homo sapiens | Apoform | X-ray | 76058 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 709 | C-c chemokine receptor type 2 | c-c chemokine receptor type 2 in complex with MTMDXAIUENDN... | ccr2_human | P41597 | Chemokine receptors | A | 6GPS | Inactive | Homo sapiens | Complex | X-ray | [(3~{s},4~{s})-3-methoxyoxan-4-yl]-[(1~{r},3~{s})-3-propan... | 60705 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 735 | C-c chemokine receptor type 2 | chimera protein of cc chemokine receptor type 2 isoform b ... | ccr2_human | P41597 | Chemokine receptors | A | 5T1A | Inactive | Homo sapiens | Complex | X-ray | Chembl4519152 Chembl3577945 | 55856 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 800 | C-c chemokine receptor type 2 | c-c chemokine receptor type 2 in complex with MTMDXAIUENDN... | ccr2_human | P41597 | Chemokine receptors | A | 6GPX | Inactive | Homo sapiens | Complex | X-ray | [(3~{s},4~{s})-3-methoxyoxan-4-yl]-[(1~{r},3~{s})-3-propan... | 61575 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 799 | C-c chemokine receptor type 2 | c-c chemokine receptor type 2 (apoform) | ccr2_human | P41597 | Chemokine receptors | A | 6GPX | Inactive | Homo sapiens | Apoform | X-ray | 61510 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 734 | C-c chemokine receptor type 2 | chimera protein of cc chemokine receptor type 2 isoform b ... | ccr2_human | P41597 | Chemokine receptors | A | 5T1A | Inactive | Homo sapiens | Apoform | X-ray | 55745 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 708 | C-c chemokine receptor type 2 | c-c chemokine receptor type 2 (apoform) | ccr2_human | P41597 | Chemokine receptors | A | 6GPS | Inactive | Homo sapiens | Apoform | X-ray | 60640 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 899 | C-c chemokine receptor type 5 | c-c chemokine receptor type 5 in complex with c-c motif ch... | ccr5_human | P51681 | Chemokine receptors | A | 5UIW | Inactive | Homo sapiens | Complex | X-ray | 84394 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1095 | C-c chemokine receptor type 5 | Chemokine Receptor CCR5 in complex with compound 21 | ccr5_human | P51681 | Chemokine receptors | A | 6AKX | Inactive | Homo sapiens | Complex | X-ray | Compound 21 | 64182 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1124 | C-c chemokine receptor type 5 | Chemokine Receptor CCR5 in complex with compound 34 | ccr5_human | P51681 | Chemokine receptors | A | 6AKY | Inactive | Homo sapiens | Complex | X-ray | Compound 34 | 67806 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 941 | C-c chemokine receptor type 5 | c-c chemokine receptor type 5 (apoform) | ccr5_human | P51681 | Chemokine receptors | A | 6AKY | Inactive | Homo sapiens | Apoform | X-ray | 67733 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 898 | C-c chemokine receptor type 5 | c-c chemokine receptor type 5 (apoform) | ccr5_human | P51681 | Chemokine receptors | A | 5UIW | Inactive | Homo sapiens | Apoform | X-ray | 71636 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 779 | C-c chemokine receptor type 5 | c-c chemokine receptor type 5 (apoform) | ccr5_human | P51681 | Chemokine receptors | A | 6AKX | Inactive | Homo sapiens | Apoform | X-ray | 64112 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 766 | Free fatty acid receptor 1 | free fatty acid receptor 1 in complex with RJZJYKXHTPUHAO-... | ffar1_human | O14842 | Free fatty acid receptors | A | 5KW2 | Active | Homo sapiens | Complex | X-ray | (3~{s})-3-cyclopropyl-3-[2-[1-[2-[2,2-dimethylpropyl-(6-me... | 54188 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 794 | Free fatty acid receptor 1 | free fatty acid receptor 1 in complex with CODQKEMYZZKQAE-... | ffar1_human | O14842 | Free fatty acid receptors | A | 5TZR | Active | Homo sapiens | Complex | X-ray | Chembl4297471 | 64914 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 929 | Free fatty acid receptor 1 | free fatty acid receptor 1 in complex with ADYYYLTWZYYGNX-... | ffar1_human | O14842 | Free fatty acid receptors | A | 5TZY | Active | Homo sapiens | Complex | X-ray | (2s,3r)-3-cyclopropyl-3-[(2r)-2-(1-{(1s)-1-[5-fluoro-2-(tr... Chembl4297471 | 59361 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 928 | Free fatty acid receptor 1 | free fatty acid receptor 1 (apoform) | ffar1_human | O14842 | Free fatty acid receptors | A | 5TZY | Active | Homo sapiens | Apoform | X-ray | 59287 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 793 | Free fatty acid receptor 1 | free fatty acid receptor 1 (apoform) | ffar1_human | O14842 | Free fatty acid receptors | A | 5TZR | Active | Homo sapiens | Apoform | X-ray | 64899 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 765 | Free fatty acid receptor 1 | free fatty acid receptor 1 (apoform) | ffar1_human | O14842 | Free fatty acid receptors | A | 5KW2 | Active | Homo sapiens | Apoform | X-ray | 54118 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 958 | Ltb4 receptor | ltb4 receptor in complex with MBLJFKQACMILLC-UHFFFAOYSA-N | q9wtk1_cavpo | Q9WTK1 | Leukotriene receptors | A | 5X33 | Inactive | Cavia porcellus | Complex | X-ray | Benzenecarboximidamide, 4-((3-((4-(1-(4-hydroxyphenyl)-1-m... | 81179 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 957 | Ltb4 receptor | ltb4 receptor (apoform) | q9wtk1_cavpo | Q9WTK1 | Leukotriene receptors | A | 5X33 | Inactive | Cavia porcellus | Apoform | X-ray | 81116 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 739 | Cysteinyl leukotriene receptor 1 | cysteinyl leukotriene receptor 1 in complex with pranlukast | cltr1_human | Q9Y271 | Leukotriene receptors | A | 6RZ4 | Active | Homo sapiens | Complex | X-ray | Azlaire | 74580 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 862 | Cysteinyl leukotriene receptor 1 | cysteinyl leukotriene receptor 1 in complex with zafirlukast | cltr1_human | Q9Y271 | Leukotriene receptors | A | 6RZ5 | Active | Homo sapiens | Complex | X-ray | Zafirlukast | 80172 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 738 | Cysteinyl leukotriene receptor 1 | cysteinyl leukotriene receptor 1 (apoform) | cltr1_human | Q9Y271 | Leukotriene receptors | A | 6RZ4 | Active | Homo sapiens | Apoform | X-ray | 74521 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 861 | Cysteinyl leukotriene receptor 1 | cysteinyl leukotriene receptor 1 (apoform) | cltr1_human | Q9Y271 | Leukotriene receptors | A | 6RZ5 | Active | Homo sapiens | Apoform | X-ray | 80055 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 691 | Hpn321 | cysteinyl leukotriene receptor 2 in complex with AXUGAYNPV... | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ9 | Active | Homo sapiens | Complex | X-ray | Ydro-1,4-benzoxazine-2-carboxylic acid | 83344 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 790 | Hpn321 | cysteinyl leukotriene receptor 2 in complex with FRDYFKGGR... | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ8 | Active | Homo sapiens | Complex | X-ray | Yl)-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid | 80329 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 806 | Hpn321 | cysteinyl leukotriene receptor 2 in complex with JCUVQOJHU... | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ7 | Active | Homo sapiens | Complex | X-ray | (2~{s})-8-[[4-[4-(2-chloranyl-5-fluoranyl-phenyl)butoxy]ph... | 70004 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 826 | Hpn321 | cysteinyl leukotriene receptor 2 in complex with JCUVQOJHU... | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ6 | Active | Homo sapiens | Complex | X-ray | (2~{s})-8-[[4-[4-(2-chloranyl-5-fluoranyl-phenyl)butoxy]ph... | 79228 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 825 | Cysteinyl leukotriene receptor 2 | cysteinyl leukotriene receptor 2 (apoform) | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ6 | Active | Homo sapiens | Apoform | X-ray | 79160 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 805 | Cysteinyl leukotriene receptor 2 | cysteinyl leukotriene receptor 2 (apoform) | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ7 | Active | Homo sapiens | Apoform | X-ray | 69972 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 789 | Cysteinyl leukotriene receptor 2 | cysteinyl leukotriene receptor 2 (apoform) | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ8 | Active | Homo sapiens | Apoform | X-ray | 80263 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 690 | Cysteinyl leukotriene receptor 2 | cysteinyl leukotriene receptor 2 (apoform) | cltr2_human | Q9NS75 | Leukotriene receptors | A | 6RZ9 | Active | Homo sapiens | Apoform | X-ray | 83294 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 871 | Lysophosphatidic acid receptor 6a | lysophosphatidic acid receptor 6a (apoform) | q08bg4_danre | Q08BG4 | Lysophospholipid (LPA) receptors | A | 5XSZ | Active | Danio rerio | Apoform | X-ray | 67298 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 897 | Cannabinoid receptor 1 | cannabinoid receptor 1 in complex with SZDVFUZKFPGYEK-WOJB... | cnr1_human | P21554 | Cannabinoid receptors | A | 5XRA | Active | Homo sapiens | Complex | X-ray | Chembl1683648 | 75000 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1002 | Cannabinoid receptor 1 | cannabinoid receptor 1 in complex with AHFZDNYNXFMRFQ-UHFF... | cnr1_human | P21554 | Cannabinoid receptors | A | 6KQI | Inactive | Homo sapiens | Complex | X-ray | Chembl559612 Chembl1553629 | 67939 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1136 | Cannabinoid receptor 1 | cannabinoid receptor 1 (apoform) | cnr1_human | P21554 | Cannabinoid receptors | A | 6KQI | Inactive | Homo sapiens | Apoform | X-ray | 67896 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 896 | Cannabinoid receptor 1 | cannabinoid receptor 1 (apoform) | cnr1_human | P21554 | Cannabinoid receptors | A | 5XRA | Active | Homo sapiens | Apoform | X-ray | 74882 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 852 | Cannabinoid receptor 1 | cannabinoid receptor 1 (apoform) | cnr1_human | P21554 | Cannabinoid receptors | A | 5XR8 | Active | Homo sapiens | Apoform | X-ray | 73955 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 956 | Cannabinoid receptor 2 | cannabinoid receptor 2 in complex with JCIYJYHFBBXSBF-HMXC... | cnr2_human | P34972 | Cannabinoid receptors | A | 6KPC | Inactive | Homo sapiens | Complex | X-ray | (6ar,9r,10ar)-9-(hydroxymethyl)-3-(8-isothiocyanato-2-meth... | 69129 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 955 | Cannabinoid receptor 2 | cannabinoid receptor 2 (apoform) | cnr2_human | P34972 | Cannabinoid receptors | A | 6KPC | Inactive | Homo sapiens | Apoform | X-ray | 69067 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 695 | Platelet-activating factor receptor | platelet-activating factor receptor in complex with GDLNHS... | ptafr_human | P25105 | Platelet-activating factor receptors | A | 5ZKQ | Active | Homo sapiens | Complex | X-ray | Abt-491 free base | 85493 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1025 | Platelet-activating factor receptor | platelet-activating factor receptor in complex with VVBFIS... | ptafr_human | P25105 | Platelet-activating factor receptors | A | 5ZKP | Other | Homo sapiens | Complex | X-ray | Foropafant | 72808 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1024 | Platelet-activating factor receptor | platelet-activating factor receptor (apoform) | ptafr_human | P25105 | Platelet-activating factor receptors | A | 5ZKP | Other | Homo sapiens | Apoform | X-ray | 72734 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 694 | Platelet-activating factor receptor | platelet-activating factor receptor (apoform) | ptafr_human | P25105 | Platelet-activating factor receptors | A | 5ZKQ | Active | Homo sapiens | Apoform | X-ray | 85436 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 885 | Prostaglandin d2 receptor 2 | prostaglandin d2 receptor 2 in complex with CANCTKXGRVNXFP... | pd2r2_human | Q9Y5Y4 | Prostanoid receptors | A | 6D27 | Inactive | Homo sapiens | Complex | X-ray | Chembl179036 | 95195 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 985 | Prostaglandin d2 receptor 2 | prostaglandin d2 receptor 2 in complex with fevipiprant | pd2r2_human | Q9Y5Y4 | Prostanoid receptors | A | 6D26 | Inactive | Homo sapiens | Complex | X-ray | Fevipiprant | 90810 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 984 | Prostaglandin d2 receptor 2 | prostaglandin d2 receptor 2 (apoform) | pd2r2_human | Q9Y5Y4 | Prostanoid receptors | A | 6D26 | Inactive | Homo sapiens | Apoform | X-ray | 90765 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 884 | Prostaglandin d2 receptor 2 | prostaglandin d2 receptor 2 (apoform) | pd2r2_human | Q9Y5Y4 | Prostanoid receptors | A | 6D27 | Inactive | Homo sapiens | Apoform | X-ray | 95145 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 749 | Prostaglandin e2 receptor ep3 subtype | prostaglandin e2 receptor ep3 subtype in complex with CNWG... | pe2r3_human | P43115 | Prostanoid receptors | A | 6M9T | Active | Homo sapiens | Complex | X-ray | (11alpha,12alpha,13e,16s)-11,16-dihydroxy-16-methyl-9-oxop... | 98305 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1027 | Prostaglandin e2 receptor ep3 subtype | prostaglandin e2 receptor ep3 subtype in complex with XEYB... | pe2r3_human | P43115 | Prostanoid receptors | A | 6AK3 | Active | Homo sapiens | Complex | X-ray | Dinoprostone | 87343 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1026 | Prostaglandin e2 receptor ep3 subtype | prostaglandin e2 receptor ep3 subtype (apoform) | pe2r3_human | P43115 | Prostanoid receptors | A | 6AK3 | Active | Homo sapiens | Apoform | X-ray | 86563 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 748 | Prostaglandin e2 receptor ep3 subtype | prostaglandin e2 receptor ep3 subtype (apoform) | pe2r3_human | P43115 | Prostanoid receptors | A | 6M9T | Active | Homo sapiens | Apoform | X-ray | 98246 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1044 | Thromboxane a2 receptor | Thromboxane A2 receptor in complex with ramatroban | ta2r_human | P21731 | Prostanoid receptors | A | 6IIU | Inactive | Homo sapiens | Complex | X-ray | Ramatroban | 85353 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1076 | Thromboxane a2 receptor | Thromboxane A2 receptor in complex with Daltroban | ta2r_human | P21731 | Prostanoid receptors | A | 6IIV | Inactive | Homo sapiens | Complex | X-ray | Daltroban | 87588 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1043 | Thromboxane a2 receptor | Thromboxane A2 receptor (apoform) | ta2r_human | P21731 | Prostanoid receptors | A | 6IIU | Inactive | Homo sapiens | Apoform | X-ray | 85301 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1075 | Thromboxane a2 receptor | Thromboxane A2 receptor (apoform) | ta2r_human | P21731 | Prostanoid receptors | A | 6IIV | Inactive | Homo sapiens | Apoform | X-ray | 87585 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 693 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME3 | Inactive | Homo sapiens | Complex | X-ray | Chembl15060 | 75024 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 713 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME2 | Inactive | Homo sapiens | Complex | X-ray | Ramelteon | 85905 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 804 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME4 | Inactive | Homo sapiens | Complex | X-ray | 2-iodomelatonin | 86671 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 808 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME5 | Inactive | Homo sapiens | Complex | X-ray | Agomelatine | 88642 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1008 | Melatonin receptor type 1a | fusion protein of melatonin receptor type 1a and glga glyc... | mtr1a_human | P48039 | Melatonin | A | 6PS8 | Inactive | Homo sapiens | Complex | X-ray | Chembl15060 | 86464 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 803 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME4 | Inactive | Homo sapiens | Apoform | X-ray | 86656 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1007 | Melatonin receptor type 1a | fusion protein of melatonin receptor type 1a and glga glyc... | mtr1a_human | P48039 | Melatonin | A | 6PS8 | Inactive | Homo sapiens | Apoform | X-ray | 86422 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 807 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME5 | Inactive | Homo sapiens | Apoform | X-ray | 88622 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 712 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME2 | Inactive | Homo sapiens | Apoform | X-ray | 85657 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 692 | Melatonin receptor type 1a | chimera protein of melatonin receptor type 1a and glga gly... | mtr1a_human | P48039 | Melatonin | A | 6ME3 | Inactive | Homo sapiens | Apoform | X-ray | 75002 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 796 | Melatonin receptor type 1b | melatonin receptor type 1b in complex with OFCLARYYBGKCHN-... | mtr1b_human | P49286 | Melatonin | A | 6ME6 | Inactive | Homo sapiens | Complex | X-ray | Chembl15060 | 76474 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 818 | Melatonin receptor type 1b | melatonin receptor type 1b in complex with YLXDSYKOBKBWJQ-... | mtr1b_human | P49286 | Melatonin | A | 6ME9 | Inactive | Homo sapiens | Complex | X-ray | Ramelteon | 65704 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 946 | Melatonin receptor type 1b | melatonin receptor type 1b in complex with OFCLARYYBGKCHN-... | mtr1b_human | P49286 | Melatonin | A | 6ME8 | Inactive | Homo sapiens | Complex | X-ray | Chembl15060 | 90412 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 994 | Melatonin receptor type 1b | melatonin receptor type 1b in complex with OFCLARYYBGKCHN-... | mtr1b_human | P49286 | Melatonin | A | 6ME7 | Inactive | Homo sapiens | Complex | X-ray | Chembl15060 | 71444 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 795 | Melatonin receptor type 1b | melatonin receptor type 1b (apoform) | mtr1b_human | P49286 | Melatonin | A | 6ME6 | Inactive | Homo sapiens | Apoform | X-ray | 76300 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 993 | Melatonin receptor type 1b | melatonin receptor type 1b (apoform) | mtr1b_human | P49286 | Melatonin | A | 6ME7 | Inactive | Homo sapiens | Apoform | X-ray | 71427 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 945 | Melatonin receptor type 1b | melatonin receptor type 1b (apoform) | mtr1b_human | P49286 | Melatonin | A | 6ME8 | Inactive | Homo sapiens | Apoform | X-ray | 90428 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 817 | Melatonin receptor type 1b | melatonin receptor type 1b (apoform) | mtr1b_human | P49286 | Melatonin | A | 6ME9 | Inactive | Homo sapiens | Apoform | X-ray | 65694 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1097 | Adenosine receptor a1 | A1 receptor in complex with PSB36 | aa1r_human | P30542 | Adenosine receptors | A | 5N2S | Inactive | Homo sapiens | Complex | X-ray | Psb36 | 95386 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 775 | Adenosine receptor a1 | adenosine receptor a1 (apoform) | aa1r_human | P30542 | Adenosine receptors | A | 5N2S | Inactive | Homo sapiens | Apoform | X-ray | 95328 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 687 | Adenosine receptor a2a | human a2a adenosine receptor t4l chimera in complex with Z... | aa2ar_human | P29274 | Adenosine receptors | A | 5WF5 | Active | Homo sapiens | Complex | X-ray | Unii-8l3oaj1r5a | 96518 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 697 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5JTB | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 96592 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 703 | Adenosine receptor a2a | adenosine receptor a2a in complex with NCWQLHHDGDXIJN-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 6GT3 | Inactive | Homo sapiens | Complex | X-ray | Chembl4594442 | 88417 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 715 | Adenosine receptor a2a | adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5OM4 | Inactive | Homo sapiens | Complex | X-ray | Chembl2024114 | 91497 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 754 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 6AQF | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 92900 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 774 | Adenosine receptor a2a | adenosine receptor a2a in complex with UJHUYWLZLDBDSR-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5UIG | Inactive | Homo sapiens | Complex | X-ray | 5-amino-n-[(2-methoxyphenyl)methyl]-2-(3-methylphenyl)-2h-... | 93865 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 784 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5NM2 | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 85353 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 814 | Adenosine receptor a2a | adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5OLZ | Inactive | Homo sapiens | Complex | X-ray | Chembl2024114 | 85035 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 828 | Adenosine receptor a2a | adenosine receptor a2a in complex with NVGMNXGIQPMJSN-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 6ZDV | Inactive | Homo sapiens | Complex | X-ray | 2-methyl-3-(4-methylthiazol-2-yl)-4-oxo-6-propyl-4h-chrome... | 90127 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 836 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5UVI | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 90205 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 854 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera in ... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2B | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 89871 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 858 | Adenosine receptor a2a | adenosine receptor a2a in complex with ZHUZHTHIEMXLRA-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5OM1 | Inactive | Homo sapiens | Complex | X-ray | Chembl2024114 | 85688 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 923 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5OLG | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 86942 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 931 | Adenosine receptor a2a | adenosine receptor a2a in complex with HQSBCDPYXDGTCL-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5OLH | Inactive | Homo sapiens | Complex | X-ray | Vipadenant | 84854 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 950 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera in ... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2D | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 83293 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 954 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5NM4 | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 86163 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 976 | Adenosine receptor a2a | adenosine receptor a2a in complex with XNBRWUQWSKXMPW-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5OLO | Inactive | Homo sapiens | Complex | X-ray | Tozadenant | 86005 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 982 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 6MH8 | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 87086 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 988 | Adenosine receptor a2a | adenosine receptor a2a in complex with CAFFEINE | aa2ar_human | P29274 | Adenosine receptors | A | 5MZP | Inactive | Homo sapiens | Complex | X-ray | Caffeine | 85190 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 992 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5NLX | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 92295 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 999 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera in ... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2C | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 84356 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1001 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 6JZH | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 102835 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1010 | Adenosine receptor a2a | human a2a adenosine receptor t4l chimera in complex with Z... | aa2ar_human | P29274 | Adenosine receptors | A | 5WF6 | Active | Homo sapiens | Complex | X-ray | Unii-8l3oaj1r5a | 115092 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1012 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5VRA | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 90122 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1014 | Adenosine receptor a2a | adenosine receptor a2a in complex with PWTBZOIUWZOPFT-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 6PS7 | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 86370 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1017 | Adenosine receptor a2a | adenosine receptor a2a in complex with KEUJAGGJGBWRFC-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 5OLV | Inactive | Homo sapiens | Complex | X-ray | Chembl1671936 | 83356 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1021 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera in ... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2A | Inactive | Homo sapiens | Complex | X-ray | Zm241385 | 94480 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1033 | Adenosine receptor a2a | adenosine receptor a2a in complex with FVMKJEVPLWCLMC-UHFF... | aa2ar_human | P29274 | Adenosine receptors | A | 6ZDR | Inactive | Homo sapiens | Complex | X-ray | Chembl2030687 | 92573 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1049 | Adenosine receptor a2a | human a2a adenosine receptor t4l chimera (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5WF5 | Active | Homo sapiens | Apoform | X-ray | Unii-8l3oaj1r5a | 96414 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 835 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5UVI | Inactive | Homo sapiens | Apoform | X-ray | Zm241385 | 90049 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1098 | Adenosine receptor a2a | A2A adenosine receptor in complex with theophylline | aa2ar_human | P29274 | Adenosine receptors | A | 5MZJ | Inactive | Homo sapiens | Complex | X-ray | Aerolate iii | 92434 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1123 | Adenosine receptor a2a | A2A adenosine receptor in complex with PSB36 | aa2ar_human | P29274 | Adenosine receptors | A | 5N2R | Inactive | Homo sapiens | Complex | X-ray | 1-butyl-3-[(~{e})-3-oxidanylprop-1-enyl]-8-[(1~{r},5~{s})-3- | 87478 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1133 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5OLV | Inactive | Homo sapiens | Apoform | X-ray | 83208 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 998 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera (ap... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2C | Inactive | Homo sapiens | Apoform | X-ray | 84200 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 991 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5NLX | Inactive | Homo sapiens | Apoform | X-ray | 92221 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 953 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5NM4 | Inactive | Homo sapiens | Apoform | X-ray | 86051 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 930 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5OLH | Inactive | Homo sapiens | Apoform | X-ray | 84705 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 857 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5OM1 | Inactive | Homo sapiens | Apoform | X-ray | 85533 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 813 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5OLZ | Inactive | Homo sapiens | Apoform | X-ray | 84899 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 753 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 6AQF | Inactive | Homo sapiens | Apoform | X-ray | 92732 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1032 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 6ZDR | Inactive | Homo sapiens | Apoform | X-ray | 92436 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1020 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera (ap... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2A | Inactive | Homo sapiens | Apoform | X-ray | 94296 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1013 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 6PS7 | Inactive | Homo sapiens | Apoform | X-ray | 86199 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1011 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5VRA | Inactive | Homo sapiens | Apoform | X-ray | 89950 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1009 | Adenosine receptor a2a | human a2a adenosine receptor t4l chimera (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5WF6 | Active | Homo sapiens | Apoform | X-ray | 114988 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1000 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 6JZH | Inactive | Homo sapiens | Apoform | X-ray | 102717 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 995 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5MZJ | Inactive | Homo sapiens | Apoform | X-ray | 92248 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 987 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5MZP | Inactive | Homo sapiens | Apoform | X-ray | 85056 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 981 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 6MH8 | Inactive | Homo sapiens | Apoform | X-ray | 87047 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 975 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5OLO | Inactive | Homo sapiens | Apoform | X-ray | 85814 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 949 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera (ap... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2D | Inactive | Homo sapiens | Apoform | X-ray | 83109 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 922 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5OLG | Inactive | Homo sapiens | Apoform | X-ray | 86745 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 906 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5N2R | Inactive | Homo sapiens | Apoform | X-ray | 87309 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 853 | Adenosine receptor a2a | adenosine receptor a2a/soluble cytochrome b562 chimera (ap... | aa2ar_human | P29274 | Adenosine receptors | A | 5K2B | Inactive | Homo sapiens | Apoform | X-ray | 89706 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 827 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 6ZDV | Inactive | Homo sapiens | Apoform | X-ray | 89993 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 783 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5NM2 | Inactive | Homo sapiens | Apoform | X-ray | 85188 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 773 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5UIG | Inactive | Homo sapiens | Apoform | X-ray | 93822 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 714 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5OM4 | Inactive | Homo sapiens | Apoform | X-ray | 91268 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 702 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 6GT3 | Inactive | Homo sapiens | Apoform | X-ray | 88265 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 696 | Adenosine receptor a2a | adenosine receptor a2a (apoform) | aa2ar_human | P29274 | Adenosine receptors | A | 5JTB | Inactive | Homo sapiens | Apoform | X-ray | 96394 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 717 | P2y purinoceptor 12 | p2y purinoceptor 12 in complex with NEMHKCNXXRQYRF-UHFFFAO... | p2y12_human | Q9H244 | P2Y receptors | A | 4NTJ | Active | Homo sapiens | Complex | X-ray | Chembl2419490 | 69106 | CLR POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 716 | P2y purinoceptor 12 | p2y purinoceptor 12 (apoform) | p2y12_human | Q9H244 | P2Y receptors | A | 4NTJ | Active | Homo sapiens | Apoform | X-ray | 69037 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 707 | Rhodopsin | rhodopsin in complex with OHAKQPWAEANPAJ-QHCPKHFHSA-N | opsd_bovin | P02699 | Opsins | A | 6FKC | Active | Bos taurus | Complex | X-ray | 3-[1'-[(2~{s})-2-(4-chlorophenyl)-3-methyl-butanoyl]spiro[... | 72963 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 721 | Rhodopsin | rhodopsin in complex with FYEGABNDKDAYPJ-UHFFFAOYSA-N | opsd_bovin | P02699 | Opsins | A | 6FKB | Active | Bos taurus | Complex | X-ray | 2-(4-chlorophenyl)-1-spiro[1,3-benzodioxole-2,4'-piperidin... | 81779 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 733 | Rhodopsin | rhodopsin in complex with QFUKMLGGPINITQ-FQEVSTJZSA-N | opsd_bovin | P02699 | Opsins | A | 6FKA | Active | Bos taurus | Complex | X-ray | (2~{s})-2-(3,4-dichlorophenyl)-3-methyl-1-spiro[1,3-benzod... | 70254 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 778 | Rhodopsin | rhodopsin in complex with RWIUNGUJHWADDD-FQEVSTJZSA-N | opsd_bovin | P02699 | Opsins | A | 6FK9 | Active | Bos taurus | Complex | X-ray | (2~{s})-3-methyl-2-phenyl-1-spiro[1,3-benzodioxole-2,4'-pi... | 71623 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 841 | Rhodopsin | rhodopsin in complex with WRVOICVPIQQYTO-LIRRHRJNSA-N | opsd_bovin | P02699 | Opsins | A | 6FK8 | Active | Bos taurus | Complex | X-ray | Haloperidol | 73974 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 913 | Rhodopsin | rhodopsin in complex with GYIGPNZLXGKQBD-KUHUBIRLSA-N | opsd_bovin | P02699 | Opsins | A | 6FK7 | Active | Bos taurus | Complex | X-ray | (2~{r},3~{r})-2-(4-chlorophenyl)-3-oxidanyl-1-spiro[1,3-be... | 72275 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 944 | Rhodopsin | rhodopsin in complex with UDAMUOKENMUCKG-FQEVSTJZSA-N | opsd_bovin | P02699 | Opsins | A | 6FK6 | Active | Bos taurus | Complex | X-ray | (2~{s})-2-(4-chlorophenyl)-3-methyl-1-spiro[1,3-benzodioxo... | 70542 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 689 | Rhodopsin | rhodopsin in complex with Lysine-Retinol | opsd_todpa | P31356 | Opsins | A | 2Z73 | Inactive | Todarodes pacificus | Complex | X-ray | N~6~-[(2z,4e,6e,8e)-3,7-dimethyl-9-(2,6,6-trimethylcyclohe... | 79918 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 757 | Rhodopsin | rhodopsin in complex with Lysine-Retinol | opsd_bovin | P02699 | Opsins | A | 3C9M | Inactive | Bos taurus | Complex | X-ray | N~6~-[(2z,4e,6e,8e)-3,7-dimethyl-9-(2,6,6-trimethylcyclohe... | 71343 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 810 | Rhodopsin | rhodopsin in complex with QLEXUFWJSPRFOP-LCYNHIKNSA-N | opsd_bovin | P02699 | Opsins | A | 5TE5 | Inactive | Bos taurus | Complex | X-ray | (2e)-{(4e)-4-[(3e)-4-(2,6,6-trimethylcyclohex-1-en-1-yl)bu... | 67530 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 873 | Rhodopsin | rhodopsin in complex with Lysine-Retinol | opsd_bovin | P02699 | Opsins | A | 5DYS | Active | Bos taurus | Complex | X-ray | N~6~-[(2z,4e,6e,8e)-3,7-dimethyl-9-(2,6,6-trimethylcyclohe... | 71625 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 895 | Rhodopsin | rhodopsin in complex with Lysine-Retinol | opsd_bovin | P02699 | Opsins | A | 1GZM | Inactive | Bos taurus | Complex | X-ray | N~6~-[(2z,4e,6e,8e)-3,7-dimethyl-9-(2,6,6-trimethylcyclohe... | 74264 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 901 | Rhodopsin | rhodopsin in complex with Lysine-Retinol | opsd_bovin | P02699 | Opsins | A | 3C9L | Inactive | Bos taurus | Complex | X-ray | N~6~-[(2z,4e,6e,8e)-3,7-dimethyl-9-(2,6,6-trimethylcyclohe... | 71307 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 943 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 6FK6 | Active | Bos taurus | Apoform | X-ray | 70431 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 912 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 6FK7 | Active | Bos taurus | Apoform | X-ray | 72216 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 809 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 5TE5 | Inactive | Bos taurus | Apoform | X-ray | 67535 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 732 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 6FKA | Active | Bos taurus | Apoform | X-ray | 70194 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 900 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 3C9L | Inactive | Bos taurus | Apoform | X-ray | 71315 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 894 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 1GZM | Inactive | Bos taurus | Apoform | X-ray | 73963 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 872 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 5DYS | Active | Bos taurus | Apoform | X-ray | 70294 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 840 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 6FK8 | Active | Bos taurus | Apoform | X-ray | 73916 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 777 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 6FK9 | Active | Bos taurus | Apoform | X-ray | 71579 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 756 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 3C9M | Inactive | Bos taurus | Apoform | X-ray | 71285 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 750 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 5TE3 | Active | Bos taurus | Apoform | X-ray | 66521 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 720 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 6FKB | Active | Bos taurus | Apoform | X-ray | 81742 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 706 | Rhodopsin | rhodopsin (apoform) | opsd_bovin | P02699 | Opsins | A | 6FKC | Active | Bos taurus | Apoform | X-ray | 72895 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 688 | Rhodopsin | rhodopsin (apoform) | opsd_todpa | P31356 | Opsins | A | 2Z73 | Inactive | Todarodes pacificus | Apoform | X-ray | 79869 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1137 | G-protein coupled receptor 52 | Chimera of G-protein coupled receptor 52 | gpr52_human | Q9Y2T5 | Class A orphans | A | 6LI0 | Inactive | Homo sapiens | Apoform | X-ray | Chembl1553629 | 111138 | POPC | 0.15 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1138 | G-protein coupled receptor 52 | Chimera of G-protein coupled receptor 52 in complex with a... | gpr52_human | Q9Y2T5 | Class A orphans | A | 6LI0 | Inactive | Homo sapiens | Complex | X-ray | Chembl4228912 | 111207 | POPC | 0.15 | ACEMD3 GPUGRID | CHARMM c36 Jul 2021 | GPCRmd community | Report |
View | 934 | G-protein coupled receptor 52 | chimera of g-protein coupled receptor 52 and flavodoxin (a... | gpr52_human | Q9Y2T5 | Class A orphans | A | 6LI1 | Inactive | Homo sapiens | Apoform | X-ray | 98239 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 986 | G-protein coupled receptor 52 | chimera of g-protein coupled receptor 52 and rubredoxin (a... | gpr52_human | Q9Y2T5 | Class A orphans | A | 6LI2 | Inactive | Homo sapiens | Apoform | X-ray | 105129 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 879 | G-protein coupled receptor homolog us28 | g-protein coupled receptor homolog us28 in complex with fr... | us28_hcmva | P69332 | Unclassified | A | 4XT3 | Active | Human cytomegalovirus (strain AD169) | Complex | X-ray | 80281 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 878 | G-protein coupled receptor homolog us28 | g-protein coupled receptor homolog us28 (apoform) | us28_hcmva | P69332 | Unclassified | A | 4XT3 | Active | Human cytomegalovirus (strain AD169) | Apoform | X-ray | 74123 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1031 | Corticotropin-releasing factor receptor 1 | corticotropin-releasing factor receptor 1 in complex with ... | crfr1_human | P34998 | Corticotropin-releasing factor receptors | B1 | 4Z9G | Inactive | Homo sapiens | Complex | X-ray | Cp-376395 | 114883 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1030 | Corticotropin-releasing factor receptor 1 | corticotropin-releasing factor receptor 1 (apoform) | crfr1_human | P34998 | Corticotropin-releasing factor receptors | B1 | 4Z9G | Inactive | Homo sapiens | Apoform | X-ray | 114829 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 699 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor in complex with MYZIDYJMN... | glp1r_human | P43220 | Glucagon receptor family | B1 | 5VEW | Inactive | Homo sapiens | Complex | X-ray | Chembl3648185 | 129085 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 705 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor in complex with MYZIDYJMN... | glp1r_human | P43220 | Glucagon receptor family | B1 | 6KK1 | Inactive | Homo sapiens | Complex | X-ray | Chembl3648185 | 128729 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 711 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor in complex with PPTKULJUD... | glp1r_human | P43220 | Glucagon receptor family | B1 | 5VEX | Inactive | Homo sapiens | Complex | X-ray | 4-{[(4-cyclohexylphenyl){[3-(methylsulfonyl)phenyl]carbamo... | 128732 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 877 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor in complex with MYZIDYJMN... | glp1r_human | P43220 | Glucagon receptor family | B1 | 6KK7 | Inactive | Homo sapiens | Complex | X-ray | Chembl3648185 | 125333 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1039 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor in complex with MYZIDYJMN... | glp1r_human | P43220 | Glucagon receptor family | B1 | 6KJV | Inactive | Homo sapiens | Complex | X-ray | Chembl3648185 | 127617 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1065 | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 (GLP-1) receptor in complex with t... | glp1r_human | P43220 | Glucagon receptor family | B1 | 5NX2 | Intermediate | Homo sapiens | Complex | X-ray | 171983 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 746 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor (apoform) | glp1r_human | P43220 | Glucagon receptor family | B1 | 6KJV | Inactive | Homo sapiens | Apoform | X-ray | 127551 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1061 | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 (GLP-1) receptor (apoform) | glp1r_human | P43220 | Glucagon receptor family | B1 | 5NX2 | Intermediate | Homo sapiens | Apoform | X-ray | 171868 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 876 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor (apoform) | glp1r_human | P43220 | Glucagon receptor family | B1 | 6KK7 | Inactive | Homo sapiens | Apoform | X-ray | 125267 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 710 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor (apoform) | glp1r_human | P43220 | Glucagon receptor family | B1 | 5VEX | Inactive | Homo sapiens | Apoform | X-ray | 128660 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 698 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor (apoform) | glp1r_human | P43220 | Glucagon receptor family | B1 | 5VEW | Inactive | Homo sapiens | Apoform | X-ray | 129019 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 704 | Glucagon-like peptide 1 receptor | glucagon-like peptide 1 receptor (apoform) | glp1r_human | P43220 | Glucagon receptor family | B1 | 6KK1 | Inactive | Homo sapiens | Apoform | X-ray | 128663 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 816 | Glucagon receptor | glucagon receptor in complex with DNTVJEMGHBIUMW-IBGZPJMES... | glr_human | P47871 | Glucagon receptor family | B1 | 5EE7 | Inactive | Homo sapiens | Complex | X-ray | Chembl1933349 | 115270 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 743 | Glucagon receptor | glucagon receptor in complex with glucagon analogue | glr_human | P47871 P01275 | Glucagon receptor family | B1 | 5YQZ | Inactive | Homo sapiens | Complex | X-ray | Pro-glucagon [cleaved into: glicentin; glicentin-related p... | 149432 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 815 | Glucagon receptor | glucagon receptor (apoform) | glr_human | P47871 | Glucagon receptor family | B1 | 5EE7 | Inactive | Homo sapiens | Apoform | X-ray | 115325 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 742 | Glucagon receptor | glucagon receptor (apoform) | glr_human | P47871 | Glucagon receptor family | B1 | 5YQZ | Inactive | Homo sapiens | Apoform | X-ray | 149058 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1135 | Parathyroid hormone/parathyroid hormone-related peptide receptor | parathyroid hormone/parathyroid hormone-related peptide re... | pth1r_human | Q03431 | Parathyroid hormone receptors | B1 | 6FJ3 | Inactive | Homo sapiens | Complex | X-ray | 152754 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 755 | Parathyroid hormone/parathyroid hormone-related peptide receptor | parathyroid hormone/parathyroid hormone-related peptide re... | pth1r_human | Q03431 | Parathyroid hormone receptors | B1 | 6FJ3 | Inactive | Homo sapiens | Apoform | X-ray | 131454 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 762 | Metabotropic glutamate receptor 5 | metabotropic glutamate receptor 5 in complex with DWPQODZA... | grm5_human | P41594 | Metabotropic glutamate receptors | C | 6FFH | Inactive | Homo sapiens | Complex | X-ray | Cid 162834 | 66219 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 843 | Metabotropic glutamate receptor 5 | metabotropic glutamate receptor 5 in complex with 2-[2-(3-... | grm5_human | P41594 | Metabotropic glutamate receptors | C | 6FFI | Inactive | Homo sapiens | Complex | X-ray | Chembl332397 | 60748 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 761 | Metabotropic glutamate receptor 5 | metabotropic glutamate receptor 5 (apoform) | grm5_human | P41594 | Metabotropic glutamate receptors | C | 6FFH | Inactive | Homo sapiens | Apoform | X-ray | 66190 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 842 | Metabotropic glutamate receptor 5 | metabotropic glutamate receptor 5 (apoform) | grm5_human | P41594 | Metabotropic glutamate receptors | C | 6FFI | Inactive | Homo sapiens | Apoform | X-ray | 60718 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 741 | Smoothened homolog | smoothened homolog in complex with ZDEZQXNVPSUJHK-UHFFFAOY... | smo_human | Q99835 | Frizzled | F | 5V57 | Inactive | Homo sapiens | Complex | X-ray | N-methyl-n-[1-[4-(2-methylpyrazol-3-yl)phthalazin-1-yl]pip... | 192748 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 772 | Smoothened homolog | smoothened homolog in complex with FOORCIAZMIWALX-JJIBRWJF... | smo_human | Q99835 | Frizzled | F | 4N4W | Inactive | Homo sapiens | Complex | X-ray | Sant-1 | 106292 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 792 | Smoothened homolog | smoothened homolog in complex with SZBGQDXLNMELTB-UHFFFAO... | smo_human | Q99835 | Frizzled | F | 4JKV | Inactive | Homo sapiens | Complex | X-ray | Taladegib | 99467 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 824 | Smoothened homolog | smoothened homolog in complex with ZDEZQXNVPSUJHK-UHFFFAOY... | smo_human | Q99835 | Frizzled | F | 5V56 | Inactive | Homo sapiens | Complex | X-ray | N-methyl-n-[1-[4-(2-methylpyrazol-3-yl)phthalazin-1-yl]pip... | 156773 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 893 | Uncharacterized protein | smoothened in complex with Cyclopamine | q98sw5_xenla | A0A1L8GTP2 | Frizzled | F | 6D32 | Active | Xenopus laevis | Complex | X-ray | 11-deoxojervine | 168207 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 933 | Smoothened homolog | smoothened homolog/soluble cytochrome b562 chimeric protei... | smo_human | Q99835 | Frizzled | F | 4QIM | Inactive | Homo sapiens | Complex | X-ray | Chembl485870 | 121012 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1023 | Smoothened homolog | smoothened homolog/soluble cytochrome b562 chimeric protei... | smo_human | Q99835 | Frizzled | F | 4O9R | Inactive | Homo sapiens | Complex | X-ray | 11-deoxojervine | 114138 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 1134 | Uncharacterized protein | smoothened in complex with CHOLESTEROL | q98sw5_xenla | A0A1L8GTP2 | Frizzled | F | 6D35 | Active | Xenopus laevis | Complex | X-ray | Cholesterol | 186024 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |
View | 791 | Smoothened homolog | smoothened homolog (apoform) | smo_human | Q99835 | Frizzled | F | 4JKV | Inactive | Homo sapiens | Apoform | X-ray | 99409 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 771 | Smoothened homolog | smoothened homolog (apoform) | smo_human | Q99835 | Frizzled | F | 4N4W | Inactive | Homo sapiens | Apoform | X-ray | 106238 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 1022 | Smoothened homolog | smoothened homolog/soluble cytochrome b562 chimeric protei... | smo_human | Q99835 | Frizzled | F | 4O9R | Inactive | Homo sapiens | Apoform | X-ray | 114068 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 932 | Smoothened homolog | smoothened homolog/soluble cytochrome b562 chimeric protei... | smo_human | Q99835 | Frizzled | F | 4QIM | Inactive | Homo sapiens | Apoform | X-ray | 120951 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 892 | Uncharacterized protein | smoothened (apoform) | q98sw5_xenla | A0A1L8GTP2 | Frizzled | F | 6D32 | Active | Xenopus laevis | Apoform | X-ray | 168091 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 888 | Uncharacterized protein | smoothened (apoform) | q98sw5_xenla | A0A1L8GTP2 | Frizzled | F | 6D35 | Active | Xenopus laevis | Apoform | X-ray | 185965 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 823 | Smoothened homolog | smoothened homolog (apoform) | smo_human | Q99835 | Frizzled | F | 5V56 | Inactive | Homo sapiens | Apoform | X-ray | 157159 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report | |
View | 740 | Smoothened homolog | smoothened homolog (apoform) | smo_human | Q99835 | Frizzled | F | 5V57 | Inactive | Homo sapiens | Apoform | X-ray | 192685 | POPC | 1.50 | ACEMD3 GPUGRID | CHARMM c36 Jul 2020 | GPCRmd community | Report |